平安! 发表于 2011-11-9 19:57 * P" b- Y$ M, t0 M$ H
Pazopanib (100 mg/kg/day free base equivalent) ' x# L* |( y2 e$ E2 H: q
这是个已经在美国上市的老药了,能下载到正式药物使用说明书英文版。6 ^ D9 U& Z- e5 y) J# U0 O
搜索了一下,原料一大堆。
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. ^$ j9 y) t7 O4 `/ Z0 p7 O2 {8 v# c对不起!100mg/kg是用于移植瘤的,我弄错了。
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以下是正版说明书的推荐用量。+ U; T7 H" L/ Z6 U! B' c( N" \
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--------------------- DOSAGE AND ADMINISTRATION ----------------
2 g: g: Z- ]( B* 800 mg orally once daily without food (at least 1 hour before or 2 hours after a meal). (2.1)
, p R& I1 y5 W: C p* Baseline moderate hepatic impairment – 200 mg orally once daily. Not recommended in patients with severe hepatic impairment. (2.2) 4 e+ t. ^! h& q9 n0 N8 f7 i( p
---------------------DOSAGE FORMS AND STRENGTHS --------------
9 n, W6 k/ H6 B7 R200 mg tablets. (3) 8 j8 C% y# I( l6 ]4 k7 x& V
-------------------------------CONTRAINDICATIONS------------------------ |